Molecule Details
InChIKeyRQBYJPVEDCXUAJ-UHFFFAOYSA-N
Compound NamePyrido(2,3-d)pyrimidine-2,4-diamine, 5-methyl-6-((methyl(5,6,7,8-tetrahydro-1-naphthalenyl)amino)methyl)-
Canonical SMILESCc1c(CN(C)c2cccc3c2CCCC3)cnc2nc(N)nc(N)c12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.56
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00374 DHFR Homo sapiens Human PF00186 6.2 IC50 ChEMBL;BindingDB
O30463 folA Mycobacterium avium Pathogen PF00186 8.7 IC50 ChEMBL
Q07422 Toxoplasma gondii Pathogen PF00186 PF00303 7.8 IC50 ChEMBL;BindingDB