Molecule Details
InChIKeyRPSFIQJOUUTWRS-UHFFFAOYSA-N
Compound Name5-(6-methoxy-7-(3-morpholinopropoxy)quinazolin-4-ylamino)-N-phenylthiophene-2-carboxamide
Canonical SMILESCOc1cc2c(Nc3ccc(C(=O)Nc4ccccc4)s3)ncnc2cc1OCCCN1CCOCC1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.72
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O14965 AURKA Homo sapiens Human PF00069 8.0 IC50 ChEMBL;BindingDB
O75716 STK16 Homo sapiens Human PF00069 8.0 pIC50 TTD_MultiTarget
Q96GD4 AURKB Homo sapiens Human PF00069 7.2 IC50 ChEMBL;BindingDB