Molecule Details
InChIKeyRPJIMTALCNCQLV-UHFFFAOYSA-N
Compound Name4-((5-(Cyclohexyloxy)(1,2,4)triazolo(1,5-A)pyrimidin-7-YL)amino)benzenesulfonamide
Canonical SMILESNS(=O)(=O)c1ccc(Nc2cc(OC3CCCCC3)nc3ncnn23)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.68
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB07688
Drug Name4-{[5-(CYCLOHEXYLOXY)[1,2,4]TRIAZOLO[1,5-A]PYRIMIDIN-7-YL]AMINO}BENZENESULFONAMIDE
CAS Numbernan
Groups experimental
ATC Codes nan
Descriptionnan

Cross-references: BindingDB: 11448 CHEMBL203407 ChemSpider: 9749376 PDB: DT5 PubChem:11574606 PubChem:99444159 ZINC: ZINC000014948097
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P06493 CDK1 Homo sapiens Human PF00069 6.8 IC50 ChEMBL;BindingDB
P49841 GSK3B Homo sapiens Human PF00069 6.7 IC50 ChEMBL
P24941 CDK2 Homo sapiens Human PF00069 6.5 pIC50 TTD_MultiTarget
DrugBank Target Actions (2)
Target Gene Target Name Action Type
P20248 CCNA2 Cyclin-A2 binder targets
P24941 CDK2 Cyclin-dependent kinase 2 binder targets