Molecule Details
InChIKeyRPGCZXUZXCJKSR-UHFFFAOYSA-N
Compound Name2-(2-azabicyclo[2.1.1]hexan-1-yl)-6-(5-methyl-1H-pyrazol-4-yl)-3H-thieno[3,2-d]pyrimidin-4-one
Canonical SMILESCc1n[nH]cc1-c1cc2nc(C34CC(CN3)C4)[nH]c(=O)c2s1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.48
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9UBU7 DBF4 Homo sapiens Human PF07535 8.7 IC50 ChEMBL;BindingDB
O00311 CDC7 Homo sapiens Human PF00069 7.1 IC50 ChEMBL;BindingDB
Q13464 ROCK1 Homo sapiens Human PF25346 PF00069 PF08912 6.7 IC50 ChEMBL;BindingDB