Molecule Details
InChIKeyROZXAOHUYCQNLS-UHFFFAOYSA-N
Compound Name5-Methoxy-6-trifluoromethyl-2,3-dihydro-indole-1-carboxylic acid pyridin-3-ylamide
Canonical SMILESCOc1cc2c(cc1C(F)(F)F)N(C(=O)Nc1cccnc1)CC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.23
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28335 HTR2C Homo sapiens Human PF00001 8.0 Ki ChEMBL;BindingDB
P05177 CYP1A2 Homo sapiens Human PF00067 7.7 IC50 ChEMBL;BindingDB
P28223 HTR2A Homo sapiens Human PF00001 6.0 Ki ChEMBL;BindingDB