Molecule Details
InChIKeyROQKQYJTPICBKQ-UHFFFAOYSA-N
Compound Name4-[4-[8-[(3-Methyl-2-pyridinyl)methyl]-2,4-dioxo-1-pyrimidin-4-yl-1,3,8-triazaspiro[4.5]decan-3-yl]phenyl]benzoic acid
Canonical SMILESCc1cccnc1CN1CCC2(CC1)C(=O)N(c1ccc(-c3ccc(C(=O)O)cc3)cc1)C(=O)N2c1ccncn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.3
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9GZT9 EGLN1 Homo sapiens Human PF13640 PF01753 9.7 IC50 ChEMBL;BindingDB
Q96KS0 EGLN2 Homo sapiens Human PF13640 9.5 IC50 ChEMBL;BindingDB
Q9H6Z9 EGLN3 Homo sapiens Human PF13640 8.7 IC50 ChEMBL;BindingDB