Molecule Details
InChIKeyRONMYLLIYUXIFC-QPJJXVBHSA-N
Compound Name(E)-3-[4-(1-methylpyrazol-4-yl)-3-pyridinyl]-N-[4-(morpholin-4-ylmethyl)phenyl]prop-2-enamide
Canonical SMILESCn1cc(-c2ccncc2/C=C/C(=O)Nc2ccc(CN3CCOCC3)cc2)cn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.07
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P24863 CCNC Homo sapiens Human PF16899 PF00134 8.2 IC50 ChEMBL;BindingDB
P49336 CDK8 Homo sapiens Human PF00069 8.2 IC50 ChEMBL
Q9BWU1 CDK19 Homo sapiens Human PF00069 7.8 IC50 ChEMBL;BindingDB