Molecule Details
InChIKeyRONKKHNZUKLQDK-UHFFFAOYSA-N
Compound Name5-[[4-[[[6,7-dimethoxy-2-(5-methylfuran-2-yl)quinolin-4-yl]amino]methyl]piperidin-1-yl]methyl]-N-hydroxythiophene-2-carboxamide
Canonical SMILESCOc1cc2nc(-c3ccc(C)o3)cc(NCC3CCN(Cc4ccc(C(=O)NO)s4)CC3)c2cc1OC
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.73
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9UBN7 HDAC6 Homo sapiens Human PF00850 PF02148 7.2 IC50 ChEMBL;BindingDB
Q13547 HDAC1 Homo sapiens Human PF00850 6.5 IC50 ChEMBL;BindingDB
P26358 DNMT1 Homo sapiens Human PF01426 PF06464 PF00145 PF12047 PF02008 6.5 IC50 ChEMBL;BindingDB