Molecule Details
InChIKeyRONFUEZMVTVAJF-VDJXWZONSA-N
Compound Name(2R,3R,4R,5S)-1-[5-[[(3S,8S,9S,10R,13R,14S,17R)-10,13-dimethyl-17-[(2R)-6-methylheptan-2-yl]-2,3,4,7,8,9,11,12,14,15,16,17-dodecahydro-1H-cyclopenta[a]phenanthren-3-yl]oxy]pentyl]-2-(hydroxymethyl)piperidine-3,4,5-triol
Canonical SMILESCC(C)CCC[C@@H](C)[C@H]1CC[C@H]2[C@@H]3CC=C4C[C@@H](OCCCCCN5C[C@H](O)[C@@H](O)[C@H](O)[C@H]5CO)CC[C@]4(C)[C@H]3CC[C@]12C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.87
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9HCG7 GBA2 Homo sapiens Human PF04685 PF12215 8.3 IC50 ChEMBL;BindingDB
P04062 GBA1 Homo sapiens Human PF02055 PF17189 6.3 IC50 ChEMBL;BindingDB
Q16739 UGCG Homo sapiens Human PF13506 6.0 IC50 ChEMBL;BindingDB