Molecule Details
InChIKeyROBGBDSQNMSQOC-LADGPHEKSA-N
Compound Name(2S,3S)-2-(4-chlorophenyl)-N-[(4-methoxyphenyl)methyl]-5-oxo-1-(4-sulfamoylphenyl)pyrrolidine-3-carboxamide
Canonical SMILESCOc1ccc(CNC(=O)[C@H]2CC(=O)N(c3ccc(S(N)(=O)=O)cc3)[C@@H]2c2ccc(Cl)cc2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.57
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00918 CA2 Homo sapiens Human PF00194 8.8 Ki ChEMBL;BindingDB
P22748 CA4 Homo sapiens Human PF00194 8.7 Ki ChEMBL;BindingDB
P43166 CA7 Homo sapiens Human PF00194 8.2 Ki ChEMBL;BindingDB