Molecule Details
InChIKeyRNWIDHFRJFXZOI-UHFFFAOYSA-N
Compound Name2-amino-N-[4-[[3-[5-(trifluoromethyl)pyridin-2-yl]oxyphenyl]methylidene]cyclohexyl]pyrimidine-5-carboxamide
Canonical SMILESNc1ncc(C(=O)NC2CCC(=Cc3cccc(Oc4ccc(C(F)(F)F)cn4)c3)CC2)cn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.59
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O00519 FAAH Homo sapiens Human PF01425 9.0 IC50 ChEMBL;BindingDB
P11712 CYP2C9 Homo sapiens Human PF00067 8.2 IC50 ChEMBL