Molecule Details
InChIKeyRNHOXGSFKJUDNY-UHFFFAOYSA-N
Compound Name4-((4-(but-2-ynyloxy)phenylsulfonyl)methyl)-N-hydroxy-1-(methylsulfonyl)piperidine-4-carboxamide
Canonical SMILESCC#CCOc1ccc(S(=O)(=O)CC2(C(=O)NO)CCN(S(C)(=O)=O)CC2)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.46
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P78536 ADAM17 Homo sapiens Human PF16698 PF00200 PF13574 8.6 IC50 ChEMBL;BindingDB
P08253 MMP2 Homo sapiens Human PF00040 PF00045 PF00413 6.3 pIC50 TTD_MultiTarget