Molecule Details
InChIKeyRLZPEQLIWYHFHH-UHFFFAOYSA-N
Compound Name4-[1-Hydroxy-1-(3-methyl-3H-imidazol-4-yl)-3-(4-pentyl-phenyl)-prop-2-ynyl]-2-naphthalen-1-yl-benzonitrile
Canonical SMILESCCCCCc1ccc(C#CC(O)(c2ccc(C#N)c(-c3cccc4ccccc34)c2)c2cncn2C)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.59
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 8.4 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 7.9 IC50 ChEMBL
P53609 PGGT1B Homo sapiens Human PF00432 6.4 IC50 ChEMBL;BindingDB