Molecule Details
InChIKeyRLPKENIQQACFGX-GOSISDBHSA-N
Compound Name(r)-2-Amino-6-borono-2-[1-(3,4-dichlorobenzyl)piperidin-4-yl]-hexanoic acid
Canonical SMILESN[C@@](CCCCB(O)O)(C(=O)O)C1CCN(Cc2ccc(Cl)c(Cl)c2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.68
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P05089 ARG1 Homo sapiens Human PF00491 7.2 IC50 ChEMBL;BindingDB
P78540 ARG2 Homo sapiens Human PF00491 6.5 IC50 ChEMBL
Q6WVP6 Schistosoma mansoni Pathogen PF00491 6.3 Kd BindingDB