Molecule Details
InChIKeyRLMPNZZDUJOQQE-UHFFFAOYSA-N
Compound Namen-(4-Chloro-3-(1h-1,2,4-triazol-5-yl)thiophen-2-yl)-2-(8-(trifluoromethyl)quinolin-5-yl)acetamide
Canonical SMILESO=C(Cc1ccc(C(F)(F)F)c2ncccc12)Nc1scc(Cl)c1-c1ncn[nH]1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.15
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P45984 MAPK9 Homo sapiens Human PF00069 7.6 IC50 ChEMBL;BindingDB
P45983 MAPK8 Homo sapiens Human PF00069 7.1 IC50 ChEMBL;BindingDB
P53779 MAPK10 Homo sapiens Human PF00069 6.7 IC50 ChEMBL;BindingDB