Molecule Details
InChIKeyRLFQVKISFLTJNU-UHFFFAOYSA-N
Compound Name2-(3-(6-isopropoxypyridin-2-yl)-1H-indol-5-yl)-5-methyl-1,3,4-oxadiazole
Canonical SMILESCc1nnc(-c2ccc3[nH]cc(-c4cccc(OC(C)C)n4)c3c2)o1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.69
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 8.0 IC50 ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 7.7 IC50 ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 7.4 IC50 ChEMBL;BindingDB