Molecule Details
InChIKeyRLDOROHJMZJOFY-CYBMUJFWSA-N
Compound Name(R)-3-bromo-5-(6-(2-(2-methylpyrrolidin-1-yl)ethyl)quinolin-2-yl)isoxazole
Canonical SMILESC[C@@H]1CCCN1CCc1ccc2nc(-c3cc(Br)no3)ccc2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.55
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9Y5N1 HRH3 Homo sapiens Human PF00001 8.7 Ki ChEMBL;BindingDB
Q12809 KCNH2 Homo sapiens Human PF00027 PF00520 PF13426 6.4 IC50 ChEMBL;BindingDB