Molecule Details
InChIKeyRKQFKAILJGXGRP-UHFFFAOYSA-N
Compound Name4-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)methyl)-7-methoxy-N-(quinuclidin-3-yl)benzofuran-2-carboxamide
Canonical SMILESCOc1cc2c(cc1OC)CN(Cc1ccc(OC)c3oc(C(=O)NC4CN5CCC4CC5)cc13)CC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.52
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P18825 ADRA2C Homo sapiens Human PF00001 9.1 Ki ChEMBL;BindingDB
P08913 ADRA2A Homo sapiens Human PF00001 7.4 Ki ChEMBL;BindingDB
P18089 ADRA2B Homo sapiens Human PF00001 6.1 Ki ChEMBL;BindingDB