Molecule Details
InChIKeyRJYKOWGBWXBBBA-AWEZNQCLSA-N
Compound Name5-[3-[4-[(3S)-3-(dimethylamino)piperidin-1-yl]pyrimidin-2-yl]-1H-indol-5-yl]-1,3,4-oxadiazol-2-amine
Canonical SMILESCN(C)[C@H]1CCCN(c2ccnc(-c3c[nH]c4ccc(-c5nnc(N)o5)cc34)n2)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.38
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9P1W9 PIM2 Homo sapiens Human PF00069 8.5 IC50 ChEMBL;BindingDB
Q86V86 PIM3 Homo sapiens Human PF00069 8.4 IC50 ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 8.2 IC50 ChEMBL;BindingDB