Molecule Details
InChIKeyRJVLFQBBRSMWHX-DHUJRADRSA-N
Compound Name4-((2S)-2-((5-Isoquinolinylsulfonyl)methylamino)-3-oxo-3-(4-phenyl-1-piperazinyl)propyl)phenyl 5-isoquinolinesulfonate
Canonical SMILESCN([C@@H](Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)C(=O)N1CCN(c2ccccc2)CC1)S(=O)(=O)c1cccc2cnccc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL6.63
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q99572 P2RX7 Homo sapiens Human PF20478 PF00864 6.8 IC50 ChEMBL;BindingDB
Q13557 CAMK2D Homo sapiens Human PF08332 PF00069 6.4 IC50 ChEMBL