Molecule Details
InChIKeyRJGDAIXCXQIWEK-UHFFFAOYSA-N
Compound Name3-[2-(8-chloro-3,4-dihydro-1H-[1]benzofuro[3,2-c]pyridin-2-yl)ethyl]-2-methylpyrido[1,2-a]pyrimidin-4-one
Canonical SMILESCc1nc2ccccn2c(=O)c1CCN1CCc2oc3ccc(Cl)cc3c2C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.69
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08913 ADRA2A Homo sapiens Human PF00001 8.4 IC50 ChEMBL;BindingDB
P18825 ADRA2C Homo sapiens Human PF00001 7.6 IC50 ChEMBL;BindingDB
P18089 ADRA2B Homo sapiens Human PF00001 7.1 IC50 ChEMBL;BindingDB