Molecule Details
InChIKeyRHPZNJJJKFQSAG-UHFFFAOYSA-N
Compound Name4-(4-(benzo[b]thiophen-2-yl)pyrimidin-2-ylamino)-N-(2-(pyrrolidin-1-yl)ethyl)benzamide
Canonical SMILESO=C(NCCN1CCCC1)c1ccc(Nc2nccc(-c3cc4ccccc4s3)n2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.32
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O14920 IKBKB Homo sapiens Human PF18397 PF12179 PF00069 6.3 IC50 ChEMBL;BindingDB
O15111 CHUK Homo sapiens Human PF18397 PF12179 PF00069 6.3 IC50 ChEMBL
Q9Y6K9 IKBKG Homo sapiens Human PF16516 PF11577 PF18414 6.3 IC50 ChEMBL