Molecule Details
InChIKeyRHFVBAXARQYYHX-UHFFFAOYSA-N
Compound Name3-(3-Carbamimidoyl-phenyl)-5-tetrazol-1-ylmethyl-4,5-dihydro-isoxazole-5-carboxylic acid (3-fluoro-2''-sulfamoyl-biphenyl-4-yl)-amide; TFA
Canonical SMILESN=C(N)c1cccc(C2=NOC(Cn3cnnn3)(C(=O)Nc3ccc(-c4ccccc4S(N)(=O)=O)cc3F)C2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.54
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00742 F10 Homo sapiens Human PF00008 PF14670 PF00594 PF00089 9.4 Ki ChEMBL;BindingDB
P07477 PRSS1 Homo sapiens Human PF00089 7.0 Ki ChEMBL;BindingDB
P00734 F2 Homo sapiens Human PF00594 PF00051 PF09396 PF00089 6.3 Ki ChEMBL;BindingDB