Molecule Details
InChIKeyRGVQQWBCJAHMTA-UHFFFAOYSA-N
Compound Name2-ethyl-3-(3-fluoro-2''-(2-cyclopropylethyloxycarbonylaminosulphonyl)-biphenyl-4-ylmethyl)-6-(N-isopropyl-N-methyl-aminocarbonylamino)-3H-quinazolin-4-one
Canonical SMILESCCc1nc2ccc(NC(=O)N(C)C(C)C)cc2c(=O)n1Cc1ccc(-c2ccccc2S(=O)(=O)NC(=O)OCCC2CC2)cc1F
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.15
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P50052 AGTR2 Homo sapiens Human PF00001 8.2 IC50 ChEMBL;BindingDB
P30556 AGTR1 Homo sapiens Human PF00001 8.1 IC50 ChEMBL;BindingDB