Molecule Details
InChIKeyRGQXJYRGDMABLT-CQSZACIVSA-N
Compound NameN-[(2R)-3-[4-(3,4-dichlorophenoxy)piperidin-1-yl]-2-hydroxypropyl]-1H-indazole-3-carboxamide
Canonical SMILESO=C(NC[C@@H](O)CN1CCC(Oc2ccc(Cl)c(Cl)c2)CC1)c1n[nH]c2ccccc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.83
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P51677 CCR3 Homo sapiens Human PF00001 8.8 Ki ChEMBL;BindingDB
P35367 HRH1 Homo sapiens Human PF00001 8.1 Ki ChEMBL;BindingDB
Q12809 KCNH2 Homo sapiens Human PF00027 PF00520 PF13426 6.6 IC50 ChEMBL;BindingDB