Molecule Details
InChIKeyRGLSQZGEAOHRTM-UHFFFAOYSA-N
Compound Name4-[1-[3-[[6-(Trifluoromethyl)pyridine-3-carbonyl]amino]phenyl]propylamino]quinazoline-8-carboxamide
Canonical SMILESCCC(Nc1ncnc2c(C(N)=O)cccc12)c1cccc(NC(=O)c2ccc(C(F)(F)F)nc2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.61
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O14965 AURKA Homo sapiens Human PF00069 9.0 IC50 ChEMBL;BindingDB
Q96GD4 AURKB Homo sapiens Human PF00069 8.8 IC50 ChEMBL;BindingDB
P23443 RPS6KB1 Homo sapiens Human PF00069 PF00433 8.0 IC50 ChEMBL;BindingDB