Molecule Details
InChIKeyRGJCMCCPAYOLOE-ZLRGZLRMSA-N
Compound NameBoc-Asp(1)-D-Tyr(SO3H)-Nle-D-Lys(1)-Trp-Nle-Asp-Phe-NH2
Canonical SMILESCCCC[C@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H]1CCCCNC(=O)C[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](Cc2ccc(OS(=O)(=O)O)cc2)C(=O)N[C@@H](CCCC)C(=O)N1)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](Cc1ccccc1)C(N)=O
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.19
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P32238 CCKAR Homo sapiens Human PF00001 PF09193 8.2 pIC50 TTD_MultiTarget
P32239 CCKBR Homo sapiens Human PF00001 8.2 Ki ChEMBL;BindingDB