Molecule Details
InChIKeyRGFGJCQSMFQBDA-GJZGRUSLSA-N
Compound Name3-[(2S,4S)-4-(4-cyanophenylmethyl)amino-2-pyrrolidinylcarbonyl]-1,3-thiazolidine
Canonical SMILESN#Cc1ccc(CN[C@@H]2CN[C@H](C(=O)N3CCSC3)C2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.59
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P27487 DPP4 Homo sapiens Human PF00930 PF00326 7.5 IC50 ChEMBL;BindingDB
Q6V1X1 DPP8 Homo sapiens Human PF19520 PF00930 PF00326 6.2 IC50 ChEMBL;BindingDB
Q86TI2 DPP9 Homo sapiens Human PF19520 PF00930 PF00326 6.1 IC50 ChEMBL;BindingDB