Molecule Details
InChIKeyRGDHGNPUKLLPLT-UHFFFAOYSA-N
Canonical SMILESO=C1CCCN1c1cc(S(=O)(=O)Nc2ccc(F)cc2F)cc2c1N(C(=O)Nc1ccc(C(F)(F)F)cc1)CC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.49
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q10469 MGAT2 Homo sapiens Human PF05060 8.5 IC50 ChEMBL;BindingDB
Q3SYC2 MOGAT2 Homo sapiens Human PF03982 8.5 IC50 ChEMBL