Molecule Details
InChIKeyREZOXLPEJRXIEV-UHFFFAOYSA-N
Compound Name5-[1-(cyclopropylmethyl)pyrazol-4-yl]-3-(6-piperazin-1-yl-2-pyridinyl)-1H-pyrazolo[3,4-c]pyridine
Canonical SMILESc1cc(-c2n[nH]c3cnc(-c4cnn(CC5CC5)c4)cc23)nc(N2CCNCC2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL10.36
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 10.8 Ki ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 10.7 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 9.6 Ki ChEMBL;BindingDB