Molecule Details
InChIKeyRERIIBOQUJUPDM-UHFFFAOYSA-N
Canonical SMILESCCC(=O)N(CC)c1cc(-c2ccc(N3CCN(C(=O)c4cc(Cc5n[nH]c(=O)c6ccccc56)ccc4F)CC3)nc2)cc(C(=O)NCc2c(C)cc(C)[nH]c2=O)c1C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.47
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q15910 EZH2 Homo sapiens Human PF21358 PF11616 PF18118 PF18264 PF00856 9.1 Kd BindingDB
Q96NZ9 PRAP1 Homo sapiens Human PF15314 7.9 IC50 ChEMBL;BindingDB