Molecule Details
InChIKeyREMZNTHJUDSMFB-UHFFFAOYSA-N
Compound Name2-anilino-4-(1H-pyrrol-3-yl) pyrimidine deriv. 8g
Canonical SMILESCc1cc(Nc2nccc(-c3c(C)[nH]c(C#N)c3C)n2)ccc1F
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.05
SourceTTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 7.0 pIC50 TTD_MultiTarget
P24941 CDK2 Homo sapiens Human PF00069 7.0 pIC50 TTD_MultiTarget