Molecule Details
InChIKeyRDXINQCCICAQJF-OQFFVEAFSA-N
Compound NameN-[4-[[(Z)-[amino-[[(4R)-4-[(2,2-diphenylacetyl)amino]-5-[(4-hydroxyphenyl)methylamino]-5-oxopentyl]amino]methylidene]carbamoyl]amino]butyl]-N'-[2-[2-[[6-[4-[[(Z)-[amino-[[(4R)-4-[(2,2-diphenylacetyl)amino]-5-[(4-hydroxyphenyl)methylamino]-5-oxopentyl]amino]methylidene]carbamoyl]amino]butylamino]-6-oxohexanoyl]amino]ethyl-(2-aminoethyl)amino]ethyl]hexanediamide
Canonical SMILESNCCN(CCNC(=O)CCCCC(=O)NCCCCNC(=O)/N=C(/N)NCCC[C@@H](NC(=O)C(c1ccccc1)c1ccccc1)C(=O)NCc1ccc(O)cc1)CCNC(=O)CCCCC(=O)NCCCCNC(=O)/N=C(/N)NCCC[C@@H](NC(=O)C(c1ccccc1)c1ccccc1)C(=O)NCc1ccc(O)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.55
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P25929 NPY1R Homo sapiens Human PF00001 7.4 Ki ChEMBL;BindingDB
P50391 NPY4R Homo sapiens Human PF00001 6.3 Ki ChEMBL;BindingDB
P49146 NPY2R Homo sapiens Human PF00001 6.0 Ki ChEMBL;BindingDB