Molecule Details
InChIKeyRDOVCRGSBIJPRK-DEOSSOPVSA-N
Compound Namebenzyl N-[(2S)-1,5-bis[(1-hydroxy-3H-2,1-benzoxaborol-6-yl)amino]-1,5-dioxopentan-2-yl]carbamate
Canonical SMILESO=C(CC[C@H](NC(=O)OCc1ccccc1)C(=O)Nc1ccc2c(c1)B(O)OC2)Nc1ccc2c(c1)B(O)OC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.93
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q16790 CA9 Homo sapiens Human PF00194 7.2 Ki ChEMBL;BindingDB
O43570 CA12 Homo sapiens Human PF00194 7.0 Ki ChEMBL;BindingDB
P00918 CA2 Homo sapiens Human PF00194 6.5 Ki ChEMBL;BindingDB