Molecule Details
InChIKeyRDECPKAPXFKZRQ-FKBYEOEOSA-N
Compound Name(S)-2-[((S)-2-{(S)-2-[2-(3H-Imidazol-4-yl)-ethylamino]-3-methyl-butyryl}-1,2,3,4-tetrahydro-isoquinoline-3-carbonyl)-amino]-4-methylsulfanyl-butyric acid
Canonical SMILESCSCC[C@H](NC(=O)[C@@H]1Cc2ccccc2CN1C(=O)[C@@H](NCCc1c[nH]cn1)C(C)C)C(=O)O
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.28
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 9.1 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 9.1 IC50 ChEMBL;BindingDB
P53609 PGGT1B Homo sapiens Human PF00432 6.6 IC50 ChEMBL