Molecule Details
InChIKeyRDAVKEYAUFGPDX-UHFFFAOYSA-N
Compound Name6,7-Dimethoxy-2-((7-methoxy-2-(2-(trifluoromethyl)phenyl)benzofuran-4-yl)methyl)-1,2,3,4-tetrahydroisoquinoline
Canonical SMILESCOc1cc2c(cc1OC)CN(Cc1ccc(OC)c3oc(-c4ccccc4C(F)(F)F)cc13)CC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.76
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P18825 ADRA2C Homo sapiens Human PF00001 7.7 Ki ChEMBL;BindingDB
P08913 ADRA2A Homo sapiens Human PF00001 6.5 Ki ChEMBL;BindingDB
P18089 ADRA2B Homo sapiens Human PF00001 6.0 Ki ChEMBL;BindingDB