Molecule Details
InChIKeyRBHCYWNSENRQLN-UHFFFAOYSA-N
Compound NamePyrazolo[1,5-b]pyridazine deriv. 45
Canonical SMILESCOc1ccc2c(-c3ccnc(Nc4ccc([N+](=O)[O-])cc4)n3)cnn2n1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.51
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 7.7 pIC50 TTD_MultiTarget
P24941 CDK2 Homo sapiens Human PF00069 7.7 pIC50 TTD_MultiTarget
P49841 GSK3B Homo sapiens Human PF00069 7.1 IC50 ChEMBL;BindingDB