Molecule Details
InChIKeyRAVPTEGGRHPKOR-UHFFFAOYSA-N
Compound Name1-[4-[4-(2-amino-4-pyridinyl)butoxy]-3-methoxyphenyl]-3-(3H-benzimidazol-5-ylmethyl)-1-(1-methylpiperidin-4-yl)urea
Canonical SMILESCOc1cc(N(C(=O)NCc2ccc3[nH]cnc3c2)C2CCN(C)CC2)ccc1OCCCCc1ccnc(N)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.33
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q16769 QPCT Homo sapiens Human PF04389 8.0 IC50 ChEMBL;BindingDB
Q9NXS2 QPCTL Homo sapiens Human PF04389 6.7 IC50 ChEMBL;BindingDB