Molecule Details
InChIKeyQZPPOPJGCFXELG-UHFFFAOYSA-N
Compound Name5-[4-(2-Hydroxy-ethyl)-piperazin-1-yl]-5-[4-(4-iodo-phenoxy)-phenyl]-pyrimidine-2,4,6-trione
Canonical SMILESO=C1NC(=O)C(c2ccc(Oc3ccc(I)cc3)cc2)(N2CCN(CCO)CC2)C(=O)N1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.43
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P14780 MMP9 Homo sapiens Human PF00040 PF00045 PF00413 8.7 IC50 ChEMBL;BindingDB
P08253 MMP2 Homo sapiens Human PF00040 PF00045 PF00413 8.2 pIC50 TTD_MultiTarget