Molecule Details
InChIKeyQYKGYRLGHZIFTF-UHFFFAOYSA-N
Compound Name2-(6-fluoro-3-((1-hydroxy-2-methylpropan-2-yl)amino)-2-methylquinoxalin-5-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one
Canonical SMILESCc1nc2ccc(F)c(-c3cc4c([nH]3)CCNC4=O)c2nc1NC(C)(C)CO
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.45
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9P1W9 PIM2 Homo sapiens Human PF00069 9.5 IC50 ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 9.0 IC50 ChEMBL;BindingDB
Q86V86 PIM3 Homo sapiens Human PF00069 6.8 IC50 ChEMBL