Molecule Details
InChIKeyQYJIOEJITUVZBJ-AWEZNQCLSA-N
Compound Name4,5,6,7-tetrahydro-1-benzothiophen-2-yl-[(3S)-3-([1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperidin-1-yl]methanone
Canonical SMILESO=C(c1cc2c(s1)CCCC2)N1CCC[C@H](c2ccnc3ncnn23)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.53
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O00408 PDE2A Homo sapiens Human PF01590 PF00233 8.0 IC50 ChEMBL;BindingDB
Q14432 PDE3A Homo sapiens Human PF00233 7.0 IC50 ChEMBL;BindingDB