Molecule Details
InChIKeyQYAUUWJPEUPHAT-UHFFFAOYSA-N
Compound Name3-bromo-N-[[2-[(7-hydroxy-6-methoxy-3,4-dihydro-1H-isoquinolin-2-yl)methyl]phenyl]methyl]benzamide
Canonical SMILESCOc1cc2c(cc1O)CN(Cc1ccccc1CNC(=O)c1cccc(Br)c1)CC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.71
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P14416 DRD2 Homo sapiens Human PF00001 6.8 Ki ChEMBL;BindingDB
P35462 DRD3 Homo sapiens Human PF00001 6.8 Ki ChEMBL;BindingDB
Q5BJF2 TMEM97 Homo sapiens Human PF05241 6.5 Ki ChEMBL;BindingDB