Molecule Details
InChIKeyQXXGDBDNPIPTRF-UHFFFAOYSA-N
Compound Name3,4-Dimethyl-7-[2-[4-[3-(1,2,3,4-tetrahydroacridin-9-ylamino)propyl]piperazin-1-yl]ethoxy]chromen-2-one
Canonical SMILESCc1c(C)c2ccc(OCCN3CCN(CCCNc4c5c(nc6ccccc46)CCCC5)CC3)cc2oc1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.12
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P22303 ACHE Homo sapiens Human PF08674 PF00135 7.8 IC50 ChEMBL;BindingDB
P06276 BCHE Homo sapiens Human PF08674 PF00135 7.0 IC50 ChEMBL;BindingDB
P27338 MAOB Homo sapiens Human PF01593 6.6 IC50 ChEMBL;BindingDB