Molecule Details
InChIKeyQXJYYBNFOZOHFW-LJQANCHMSA-N
Compound Name5-chloro-2-fluoro-4-[[(6S)-5-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-6-yl]methylamino]-N-(1,3-thiazol-2-yl)benzenesulfonamide
Canonical SMILESO=S(=O)(Nc1nccs1)c1cc(Cl)c(NC[C@H]2NCCC=C2c2ccc(F)cc2)cc1F
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.13
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q15858 SCN9A Homo sapiens Human PF00520 PF24609 PF06512 PF11933 7.5 IC50 ChEMBL;BindingDB
P11712 CYP2C9 Homo sapiens Human PF00067 7.5 IC50 ChEMBL;BindingDB
P33261 CYP2C19 Homo sapiens Human PF00067 6.4 IC50 ChEMBL;BindingDB