Molecule Details
InChIKeyQXEZLMVQNMVYRX-UHFFFAOYSA-N
Compound Name7-Bromo-9,10-dihydro-phenanthrene-2-carboxylic acid
Canonical SMILESO=C(O)c1ccc2c(c1)CCc1cc(Br)ccc1-2
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.59
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 7.6 pIC50 TTD_MultiTarget
P31639 SLC5A2 Homo sapiens Human PF00474 7.6 pIC50 TTD_MultiTarget
P18405 SRD5A1 Homo sapiens Human PF02544 7.6 Ki ChEMBL;BindingDB