Molecule Details
InChIKeyQWRCKPSAXDHLDB-PVTUVMIMSA-N
Compound Name(2S)-2-amino-N-[4-[(2S,5S,8S,14S,17R)-8,14-dibenzyl-5-[(1R)-1-hydroxyethyl]-17-(1H-indol-3-ylmethyl)-3,6,9,12,15,18-hexaoxo-10-[(1R)-1-phenylethyl]-1,4,7,10,13,16-hexazacyclooctadec-2-yl]butyl]-3-phenylpropanamide
Canonical SMILESC[C@H](c1ccccc1)N1CC(=O)N[C@@H](Cc2ccccc2)C(=O)N[C@H](Cc2c[nH]c3ccccc23)C(=O)N[C@@H](CCCCNC(=O)[C@@H](N)Cc2ccccc2)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](Cc2ccccc2)C1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.34
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P30874 SSTR2 Homo sapiens Human PF00001 8.6 Kd ChEMBL;BindingDB
P35346 SSTR5 Homo sapiens Human PF00001 7.0 Kd ChEMBL;BindingDB
P32745 SSTR3 Homo sapiens Human PF00001 6.4 Kd ChEMBL;BindingDB