Molecule Details
InChIKeyQWCWGAZSLRLOPF-UHFFFAOYSA-N
Compound Name5-[3-[6-(3-methyl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)-2-pyridinyl]-1H-indol-5-yl]-1,3,4-thiadiazol-2-amine
Canonical SMILESCc1nnc2n1CCN(c1cccc(-c3c[nH]c4ccc(-c5nnc(N)s5)cc34)n1)C2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.78
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 8.5 IC50 ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 7.8 IC50 ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 7.0 IC50 ChEMBL;BindingDB