Molecule Details
InChIKeyQVUNFYOXAPUVEZ-UHFFFAOYSA-N
Compound Name4-benzylsulfanyl-2-oxo-5,6-dihydro-3H-benzo[f]isoquinoline-1-carbonitrile
Canonical SMILESN#Cc1c(O)nc(SCc2ccccc2)c2c1-c1ccccc1CC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.36
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P28845 HSD11B1 Homo sapiens Human PF00106 8.3 IC50 ChEMBL;BindingDB
P80365 HSD11B2 Homo sapiens Human PF00106 6.4 IC50 ChEMBL;BindingDB