Molecule Details
InChIKeyQVQWCYWOMABSFT-MPQUPPDSSA-N
Compound Name(18S,21R)-21-(benzylsulfonylamino)-N-[(4-carbamimidoylphenyl)methyl]-3,10,20-trioxo-2,5,8,11,19-pentazatetracyclo[21.2.2.25,8.112,16]triaconta-1(26),12,14,16(28),23(27),24-hexaene-18-carboxamide
Canonical SMILESN=C(N)c1ccc(CNC(=O)[C@@H]2Cc3cccc(c3)NC(=O)CN3CCN(CC3)CC(=O)Nc3ccc(cc3)C[C@@H](NS(=O)(=O)Cc3ccccc3)C(=O)N2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.74
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P03952 KLKB1 Homo sapiens Human PF00024 PF00089 7.9 Ki ChEMBL;BindingDB
P00747 PLG Homo sapiens Human PF00051 PF00024 PF00089 7.6 Ki ChEMBL;BindingDB