Molecule Details
InChIKeyQVLFTJGCGVDBFK-LYASGPROSA-N
Compound NameN(1)His-D-2Nal-Arg-D-Trp-D-Lys(2)-NH2.Ac-Nle-D-Asp(1)-(2)
Canonical SMILESCCCC[C@H](NC(C)=O)C(=O)N[C@@H]1CC(=O)N[C@@H](Cc2c[nH]cn2)C(=O)N[C@H](Cc2ccc3ccccc3c2)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@H](Cc2c[nH]c3ccccc23)C(=O)N[C@@H](C(N)=O)CCCCNC1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.05
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P32245 MC4R Homo sapiens Human PF00001 9.1 Ki ChEMBL;BindingDB
P33032 MC5R Homo sapiens Human PF00001 7.5 Ki ChEMBL;BindingDB
P41968 MC3R Homo sapiens Human PF00001 7.5 Ki ChEMBL;BindingDB